serw-MX  [xml]  
 


    
 DeCS Categories

D03 Heterocyclic Compounds .
D03.132 Alkaloids .
D03.132.577 Opiate Alkaloids .
D03.132.577.249 Morphinans .
D03.132.577.249.106 Benzomorphans .
D03.132.577.249.106.700 Pentazocine .
D03.132.577.249.150 Buprenorphine .
D03.132.577.249.606 Nalbuphine .
D03.132.577.249.656 Nalorphine .
D03.132.577.249.706 Naloxone .
D03.605 Heterocyclic Compounds, Bridged-Ring .
D03.605.497 Morphinans .
D03.605.497.150 Buprenorphine .
D03.605.497.639 Nalbuphine .
D03.605.497.694 Nalorphine .
D03.605.497.750 Naloxone .
D03.633 Heterocyclic Compounds, Fused-Ring .
D03.633.400 Heterocyclic Compounds, 4 or More Rings .
D03.633.400.686 Morphinans .
D03.633.400.686.150 Buprenorphine .
D03.633.400.686.639 Nalbuphine .
D03.633.400.686.694 Nalorphine .
D03.633.400.686.750 Naloxone .
D04 Polycyclic Compounds .
D04.615 Polycyclic Aromatic Hydrocarbons .
D04.615.723 Phenanthrenes .
D04.615.723.795 Morphinans .
D04.615.723.795.106 Benzomorphans .
D04.615.723.795.106.700 Pentazocine .
D04.615.723.795.150 Buprenorphine .
D04.615.723.795.606 Nalbuphine .
D04.615.723.795.656 Nalorphine .
D04.615.723.795.706 Naloxone .
D27 Chemical Actions and Uses .
D27.505 Pharmacologic Actions .
D27.505.696 Physiological Effects of Drugs .
D27.505.696.277 Central Nervous System Depressants .
D27.505.696.277.600 Narcotics .
D27.505.696.277.600.500 Analgesics, Opioid .
D27.505.696.663 Peripheral Nervous System Agents .
D27.505.696.663.850 Sensory System Agents .
D27.505.696.663.850.014 Analgesics .
D27.505.696.663.850.014.760 Narcotics .
D27.505.696.663.850.014.760.500 Analgesics, Opioid .
D27.505.954 Therapeutic Uses .
D27.505.954.427 Central Nervous System Agents .
D27.505.954.427.040 Analgesics .
D27.505.954.427.040.550 Narcotics .
D27.505.954.427.040.550.500 Analgesics, Opioid .
D27.505.954.427.210 Central Nervous System Depressants .
D27.505.954.427.210.600 Narcotics .
D27.505.954.427.210.600.500 Analgesics, Opioid .
 
 Terms
 Synonyms & Historicals
Documents
LILACS e MDL
 
Buprenorphine .
6029-M .
Buprenex .
Buprenorphine Hydrochloride .
Buprex .
Prefin .
RX-6029-M .
Subutex .
Temgesic .
Temgésic .
6029 M .
6029M .
Hydrochloride, Buprenorphine .
RX 6029 M .
RX6029M .
A derivative of the opioid alkaloid THEBAINE that is a more potent and longer lasting analgesic than MORPHINE. It appears to act as a partial agonist at mu and kappa opioid receptors and as an antagonist at delta receptors. The lack of delta-agonist activity has been suggested to account for the observation that buprenorphine tolerance may not develop with chronic use. .
1.00
604392
 
Naloxone .
MRZ 2593-Br .
MRZ-2593 .
Nalone .
Naloxon Curamed .
Naloxon-Ratiopharm .
Naloxone Abello .
Naloxone Hydrobromide .
Naloxone Hydrochloride .
Naloxone Hydrochloride Dihydride .
Naloxone Hydrochloride, (5 beta,9 alpha,13 alpha,14 alpha)-Isomer .
Naloxone, (5 beta,9 alpha,13 alpha,14 alpha)-Isomer .
Narcan .
Narcanti .
Abello, Naloxone .
Curamed, Naloxon .
Dihydride, Naloxone Hydrochloride .
Hydrobromide, Naloxone .
Hydrochloride Dihydride, Naloxone .
Hydrochloride, Naloxone .
MRZ 2593 .
MRZ 2593 Br .
MRZ 2593Br .
MRZ2593 .
Naloxon Ratiopharm .
A specific opiate antagonist that has no agonist activity. It is a competitive antagonist at mu, delta, and kappa opioid receptors. .
0.56
10317915
 
Nalbuphine .
EN-2234A .
Nalbuphine Hydrochloride .
Nalbuphine Serb .
Nubain .
EN 2234A .
EN2234A .
Hydrochloride, Nalbuphine .
A narcotic used as a pain medication. It appears to be an agonist at kappa opioid receptors and an antagonist or partial agonist at mu opioid receptors. .
0.54
53636
 
Pentazocine .
Fortral .
Lexir .
Pentazocine Hydrochloride .
Pentazocine Lactate .
Talwin .
Hydrochloride, Pentazocine .
Lactate, Pentazocine .
The first mixed agonist-antagonist analgesic to be marketed. It is an agonist at the kappa and sigma opioid receptors and has a weak antagonist action at the mu receptor. (From AMA Drug Evaluations Annual, 1991, p97) .
0.49
42183
 
Nalorphine .
Lethidrone .
Nalorphine Hydrobromide .
Nalorphine Hydrochloride .
Nalorphine, (14 alpha)-Isomer .
Nalorphine, L-tartrate (1:1) .
Hydrobromide, Nalorphine .
Hydrochloride, Nalorphine .
Allylnormorphine .
A narcotic antagonist with some agonist properties. It is an antagonist at mu opioid receptors and an agonist at kappa opioid receptors. Given alone it produces a broad spectrum of unpleasant effects and it is considered to be clinically obsolete. .
0.49
2801
 
Analgesics, Opioid .
Full Opioid Agonists .
Opioid Full Agonists .
Opioid Mixed Agonist-Antagonists .
Opioid Partial Agonists .
Partial Opioid Agonists .
Agonist-Antagonists, Opioid Mixed .
Agonists, Full Opioid .
Agonists, Opioid Full .
Agonists, Opioid Partial .
Agonists, Partial Opioid .
Full Agonists, Opioid .
Mixed Agonist-Antagonists, Opioid .
Opioid Agonists, Full .
Opioid Agonists, Partial .
Opioid Mixed Agonist Antagonists .
Partial Agonists, Opioid .
Opioid Analgesics .
Opioids .
Analgesics, Addictive .
Compounds with activity like OPIATE ALKALOIDS, acting at OPIOID RECEPTORS. Properties include induction of ANALGESIA or NARCOSIS. .
0.41
44535259