serw-MX  [xml]  
 


    
 DeCS Categories

D03 Heterocyclic Compounds .
D03.132 Alkaloids .
D03.132.577 Opiate Alkaloids .
D03.132.577.249 Morphinans .
D03.132.577.249.106 Benzomorphans .
D03.132.577.249.106.700 Pentazocine .
D03.132.577.249.150 Buprenorphine .
D03.132.577.249.606 Nalbuphine .
D03.132.577.249.656 Nalorphine .
D03.132.577.249.706 Naloxone .
D03.605 Heterocyclic Compounds, Bridged-Ring .
D03.605.497 Morphinans .
D03.605.497.150 Buprenorphine .
D03.605.497.639 Nalbuphine .
D03.605.497.694 Nalorphine .
D03.605.497.750 Naloxone .
D03.633 Heterocyclic Compounds, Fused-Ring .
D03.633.400 Heterocyclic Compounds, 4 or More Rings .
D03.633.400.686 Morphinans .
D03.633.400.686.150 Buprenorphine .
D03.633.400.686.639 Nalbuphine .
D03.633.400.686.694 Nalorphine .
D03.633.400.686.750 Naloxone .
D04 Polycyclic Compounds .
D04.615 Polycyclic Aromatic Hydrocarbons .
D04.615.723 Phenanthrenes .
D04.615.723.795 Morphinans .
D04.615.723.795.106 Benzomorphans .
D04.615.723.795.106.700 Pentazocine .
D04.615.723.795.150 Buprenorphine .
D04.615.723.795.606 Nalbuphine .
D04.615.723.795.656 Nalorphine .
D04.615.723.795.706 Naloxone .
D06 Hormones, Hormone Substitutes, and Hormone Antagonists .
D06.347 Hormone Antagonists .
D06.347.065 Androgen Antagonists .
D06.347.065.249 Androgen Receptor Antagonists .
D27 Chemical Actions and Uses .
D27.505 Pharmacologic Actions .
D27.505.696 Physiological Effects of Drugs .
D27.505.696.277 Central Nervous System Depressants .
D27.505.696.277.600 Narcotics .
D27.505.696.277.600.500 Analgesics, Opioid .
D27.505.696.399 Hormones, Hormone Substitutes, and Hormone Antagonists .
D27.505.696.399.450 Hormone Antagonists .
D27.505.696.399.450.065 Androgen Antagonists .
D27.505.696.399.450.065.249 Androgen Receptor Antagonists .
D27.505.696.399.472 Hormones .
D27.505.696.399.472.161 Androgens .
D27.505.696.663 Peripheral Nervous System Agents .
D27.505.696.663.850 Sensory System Agents .
D27.505.696.663.850.014 Analgesics .
D27.505.696.663.850.014.760 Narcotics .
D27.505.696.663.850.014.760.500 Analgesics, Opioid .
D27.505.954 Therapeutic Uses .
D27.505.954.427 Central Nervous System Agents .
D27.505.954.427.040 Analgesics .
D27.505.954.427.040.550 Narcotics .
D27.505.954.427.040.550.500 Analgesics, Opioid .
D27.505.954.427.210 Central Nervous System Depressants .
D27.505.954.427.210.600 Narcotics .
D27.505.954.427.210.600.500 Analgesics, Opioid .
 
 Terms
 Synonyms & Historicals
Documents
LILACS e MDL
 
Pentazocine .
Fortral .
Lexir .
Pentazocine Hydrochloride .
Pentazocine Lactate .
Talwin .
Hydrochloride, Pentazocine .
Lactate, Pentazocine .
The first mixed agonist-antagonist analgesic to be marketed. It is an agonist at the kappa and sigma opioid receptors and has a weak antagonist action at the mu receptor. (From AMA Drug Evaluations Annual, 1991, p97) .
1.00
42183
 
Nalbuphine .
EN-2234A .
Nalbuphine Hydrochloride .
Nalbuphine Serb .
Nubain .
EN 2234A .
EN2234A .
Hydrochloride, Nalbuphine .
A narcotic used as a pain medication. It appears to be an agonist at kappa opioid receptors and an antagonist or partial agonist at mu opioid receptors. .
0.59
53636
 
Naloxone .
MRZ 2593-Br .
MRZ-2593 .
Nalone .
Naloxon Curamed .
Naloxon-Ratiopharm .
Naloxone Abello .
Naloxone Hydrobromide .
Naloxone Hydrochloride .
Naloxone Hydrochloride Dihydride .
Naloxone Hydrochloride, (5 beta,9 alpha,13 alpha,14 alpha)-Isomer .
Naloxone, (5 beta,9 alpha,13 alpha,14 alpha)-Isomer .
Narcan .
Narcanti .
Abello, Naloxone .
Curamed, Naloxon .
Dihydride, Naloxone Hydrochloride .
Hydrobromide, Naloxone .
Hydrochloride Dihydride, Naloxone .
Hydrochloride, Naloxone .
MRZ 2593 .
MRZ 2593 Br .
MRZ 2593Br .
MRZ2593 .
Naloxon Ratiopharm .
A specific opiate antagonist that has no agonist activity. It is a competitive antagonist at mu, delta, and kappa opioid receptors. .
0.56
10317915
 
Nalorphine .
Lethidrone .
Nalorphine Hydrobromide .
Nalorphine Hydrochloride .
Nalorphine, (14 alpha)-Isomer .
Nalorphine, L-tartrate (1:1) .
Hydrobromide, Nalorphine .
Hydrochloride, Nalorphine .
Allylnormorphine .
A narcotic antagonist with some agonist properties. It is an antagonist at mu opioid receptors and an agonist at kappa opioid receptors. Given alone it produces a broad spectrum of unpleasant effects and it is considered to be clinically obsolete. .
0.54
2801
 
Buprenorphine .
6029-M .
Buprenex .
Buprenorphine Hydrochloride .
Buprex .
Prefin .
RX-6029-M .
Subutex .
Temgesic .
Temgésic .
6029 M .
6029M .
Hydrochloride, Buprenorphine .
RX 6029 M .
RX6029M .
A derivative of the opioid alkaloid THEBAINE that is a more potent and longer lasting analgesic than MORPHINE. It appears to act as a partial agonist at mu and kappa opioid receptors and as an antagonist at delta receptors. The lack of delta-agonist activity has been suggested to account for the observation that buprenorphine tolerance may not develop with chronic use. .
0.49
604392
 
Androgen Receptor Antagonists .
Antagonists, Androgen Receptor .
Receptor Antagonists, Androgen .
Compounds that bind to and inhibit the activation of ANDROGEN RECEPTORS. .
0.48
01050
 
Androgens .
Androgen Effect .
Androgen Effects .
Androgen Receptor Agonists .
Androgenic Agents .
Androgenic Compounds .
Agents, Androgenic .
Agonists, Androgen Receptor .
Compounds, Androgenic .
Effect, Androgen .
Effects, Androgen .
Receptor Agonists, Androgen .
Compounds that interact with ANDROGEN RECEPTORS in target tissues to bring about the effects similar to those of TESTOSTERONE. Depending on the target tissues, androgenic effects can be on SEX DIFFERENTIATION; male reproductive organs, SPERMATOGENESIS; secondary male SEX CHARACTERISTICS; LIBIDO; development of muscle mass, strength, and power. .
0.48
28622358
 
Analgesics, Opioid .
Full Opioid Agonists .
Opioid Full Agonists .
Opioid Mixed Agonist-Antagonists .
Opioid Partial Agonists .
Partial Opioid Agonists .
Agonist-Antagonists, Opioid Mixed .
Agonists, Full Opioid .
Agonists, Opioid Full .
Agonists, Opioid Partial .
Agonists, Partial Opioid .
Full Agonists, Opioid .
Mixed Agonist-Antagonists, Opioid .
Opioid Agonists, Full .
Opioid Agonists, Partial .
Opioid Mixed Agonist Antagonists .
Partial Agonists, Opioid .
Opioid Analgesics .
Opioids .
Analgesics, Addictive .
Compounds with activity like OPIATE ALKALOIDS, acting at OPIOID RECEPTORS. Properties include induction of ANALGESIA or NARCOSIS. .
0.47
45235259